Molecule Details
InChIKeyFTXAKSJEBVGKHR-HDICACEKSA-N
Canonical SMILESCOc1cc(OC)cc(C(=O)N[C@H]2CC[C@@H](Nc3nc(N(C)C)c4ccccc4n3)CC2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.92
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q99705 MCHR1 Homo sapiens Human PF00001 8.7 IC50 ChEMBL;BindingDB
P08913 ADRA2A Homo sapiens Human PF00001 7.2 IC50 ChEMBL;BindingDB