Molecule Details
InChIKeyFTQDJVZNPJRVPG-XWEVEMRCSA-N
Canonical SMILESCC(=O)O[C@H]1CC[C@]2(C)[C@H]3C(=O)C=C4[C@@H]5C[C@@](C)(C(=O)O)CC[C@]5(C)CC[C@@]4(C)[C@]3(C)CC[C@H]2C1(C)C
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.11
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
DrugBank Annotations
DrugBank ID DB13640
Drug NameAcetoxolone
CAS Number6277-14-1
Groups experimental
ATC Codes A02BX09
Descriptionnan

Categories: Alimentary Tract and Metabolism Drugs for Acid Related Disorders Drugs for Peptic Ulcer and Gastro-Oesophageal Reflux Disease (Gord) Pentacyclic Triterpenes Terpenes Triterpenes
Cross-references: BindingDB: 50188385 ChEBI: 81306 CHEMBL207413 ChemSpider: 85123 C17734 RxCUI: 16784 Wikipedia: Acetoxolone ZINC: ZINC000034169081
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P80365 HSD11B2 Homo sapiens Human PF00106 6.1 IC50 ChEMBL;BindingDB
P28845 HSD11B1 Homo sapiens Human PF00106 6.1 IC50 ChEMBL;BindingDB