Molecule Details
InChIKeyFTHLNVOKHACXIU-HXUWFJFHSA-N
Compound Name(4R)-4-(4-chlorophenyl)-2-cyclopropyl-5-(1,5-dimethyl-6-oxo-3-pyridinyl)-3-methyl-4H-pyrrolo[3,4-c]pyrazol-6-one
Canonical SMILESCc1cc(N2C(=O)c3nn(C4CC4)c(C)c3[C@H]2c2ccc(Cl)cc2)cn(C)c1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.34
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q15059 BRD3 Homo sapiens Human PF17035 PF00439 7.4 IC50 ChEMBL;BindingDB
O60885 BRD4 Homo sapiens Human PF17035 PF17105 PF00439 7.3 IC50 ChEMBL;BindingDB
P25440 BRD2 Homo sapiens Human PF17035 PF00439 7.3 IC50 ChEMBL;BindingDB