Molecule Details
InChIKeyFTBVOTPFSOMUEE-UHFFFAOYSA-N
Compound Name1-cyclopentyl-3-[7-(1H-pyrazol-4-yl)pyrido[3,2-d]pyrimidin-2-yl]urea
Canonical SMILESO=C(Nc1ncc2ncc(-c3cn[nH]c3)cc2n1)NC1CCCC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.56
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P42338 PIK3CB Homo sapiens Human PF00454 PF00792 PF02192 PF00794 PF00613 8.3 IC50 ChEMBL
P42336 PIK3CA Homo sapiens Human PF00454 PF00792 PF02192 PF00794 PF00613 7.2 IC50 ChEMBL
P28482 MAPK1 Homo sapiens Human PF00069 7.1 IC50 ChEMBL