Molecule Details
InChIKeyFSSFYFUDWJPZMF-UHFFFAOYSA-N
Compound Name1-Methyl-2-oxo-5-[3-(trifluoromethoxy)phenyl]-6-[alpha-(1-methyl-1H-imidazole-5-yl)-4-cyanobenzyloxymethyl]-1,2-dihydropyridine-3-carbonitrile
Canonical SMILESCn1cncc1C(OCc1c(-c2cccc(OC(F)(F)F)c2)cc(C#N)c(=O)n1C)c1ccc(C#N)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL9.38
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 9.4 pIC50 TTD_MultiTarget
P49356 FNTB Homo sapiens Human PF00432 9.4 IC50 ChEMBL