Molecule Details
InChIKeyFSRCBTSVLQDXOV-UHFFFAOYSA-N
Compound Name8-(3-Nitro-phenyl)-6-pyridin-3-yl-[1,7]naphthyridine
Canonical SMILESO=[N+]([O-])c1cccc(-c2nc(-c3cccnc3)cc3cccnc23)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.22
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q08499 PDE4D Homo sapiens Human PF18100 PF00233 8.5 IC50 ChEMBL;BindingDB
P27815 PDE4A Homo sapiens Human PF18100 PF00233 6.9 IC50 ChEMBL;BindingDB
Q08493 PDE4C Homo sapiens Human PF18100 PF00233 6.2 IC50 ChEMBL;BindingDB