Molecule Details
InChIKeyFSLWZIRTOUAUNP-UHFFFAOYSA-N
Compound Name8-Hydroxy-5-[4-(4-pyrazolo[1,5-a]pyridin-5-yloxybutyl)piperazin-1-yl]chromen-2-one
Canonical SMILESO=c1ccc2c(N3CCN(CCCCOc4ccn5nccc5c4)CC3)ccc(O)c2o1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.4
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P35462 DRD3 Homo sapiens Human PF00001 8.1 Ki ChEMBL;BindingDB
P14416 DRD2 Homo sapiens Human PF00001 7.6 Ki ChEMBL;BindingDB
P21917 DRD4 Homo sapiens Human PF00001 6.6 Ki ChEMBL;BindingDB