Molecule Details
InChIKeyFRKWBPZUTQTJCZ-UHFFFAOYSA-N
Compound Name4-ethyl-N-[2-[4-[[2-ethyl-4-oxo-6-(propan-2-ylcarbamoylamino)quinazolin-3-yl]methyl]-3-fluorophenyl]phenyl]sulfonyl-2-fluorobenzamide
Canonical SMILESCCc1ccc(C(=O)NS(=O)(=O)c2ccccc2-c2ccc(Cn3c(CC)nc4ccc(NC(=O)NC(C)C)cc4c3=O)c(F)c2)c(F)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.66
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P30556 AGTR1 Homo sapiens Human PF00001 8.8 IC50 ChEMBL;BindingDB
P50052 AGTR2 Homo sapiens Human PF00001 8.5 IC50 ChEMBL;BindingDB