Molecule Details
InChIKeyFRKIPPLTMSQJLF-UHFFFAOYSA-N
Compound Name3-(4-Fluorophenyl)-5-(4-(4-methyl-5-(2-(trifluoromethyl)phenyl)-4H-1,2,4-triazol-3-yl)bicyclo(2.2.2)octan-1-yl)-1,2,4-oxadiazole
Canonical SMILESCn1c(-c2ccccc2C(F)(F)F)nnc1C12CCC(c3nc(-c4ccc(F)cc4)no3)(CC1)CC2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.61
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P14061 HSD17B1 Homo sapiens Human PF00106 8.7 IC50 ChEMBL;BindingDB
P28845 HSD11B1 Homo sapiens Human PF00106 8.7 IC50 ChEMBL;BindingDB
P80365 HSD11B2 Homo sapiens Human PF00106 8.5 IC50 ChEMBL;BindingDB