Molecule Details
InChIKeyFRJJESBRJAYWNY-UHFFFAOYSA-O
Compound Name1-[(2,3-Dichloro-4,6-disulfamoyl-phenylcarbamoyl)-methyl]-2,4,6-trimethyl-pyridinium; perchlorate
Canonical SMILESCc1cc(C)[n+](CC(=O)Nc2c(S(N)(=O)=O)cc(S(N)(=O)=O)c(Cl)c2Cl)c(C)c1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.25
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00918 CA2 Homo sapiens Human PF00194 7.7 Ki ChEMBL;BindingDB
P18505 GABRB1 Homo sapiens Human PF02931 PF02932 7.7 pIC50 TTD_MultiTarget
P00915 CA1 Homo sapiens Human PF00194 6.3 Ki ChEMBL;BindingDB