Molecule Details
InChIKeyFRDOLUJNVQSLJJ-UHFFFAOYSA-N
Canonical SMILESCOc1cc(CN2CCN(c3ccccc3OC)CC2)ccc1OCc1cn(CCCCCCCCN(C)CCCCCNC(=O)COc2cccc(C#Cc3csc(C)n3)c2)nn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL6.78
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P14416 DRD2 Homo sapiens Human PF00001 6.9 Ki ChEMBL;BindingDB
P41594 GRM5 Homo sapiens Human PF00003 PF01094 PF10606 PF07562 6.6 IC50 ChEMBL;BindingDB