Molecule Details
InChIKeyFQZYFIYBPFXEFC-UHFFFAOYSA-N
Compound Namemethyl 2-[4-(1-cyclooctylpiperidin-4-yl)-3-oxoquinoxalin-2-yl]-3,4-dihydro-1H-isoquinoline-7-carboxylate
Canonical SMILESCOC(=O)c1ccc2c(c1)CN(c1nc3ccccc3n(C3CCN(C4CCCCCCC4)CC3)c1=O)CC2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.59
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q5TC84 OGFRL1 Homo sapiens Human PF04664 7.0 Ki ChEMBL;BindingDB
P41145 OPRK1 Homo sapiens Human PF00001 6.5 Ki ChEMBL;BindingDB
P35372 OPRM1 Homo sapiens Human PF00001 6.3 Ki ChEMBL;BindingDB