Molecule Details
InChIKeyFQVJSQJPMQVZKV-UHFFFAOYSA-N
Compound Name3-{3-[5-(morpholin-4-ylmethyl)-1H-1,3-benzodiazol-2-yl]-1H-pyrazol-4-yl}-1-oxan-4-ylurea
Canonical SMILESO=C(Nc1c[nH]nc1-c1nc2cc(CN3CCOCC3)ccc2[nH]1)NC1CCOCC1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.72
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q96GD4 AURKB Homo sapiens Human PF00069 8.0 IC50 ChEMBL;BindingDB
O75716 STK16 Homo sapiens Human PF00069 7.6 pIC50 TTD_MultiTarget
O14965 AURKA Homo sapiens Human PF00069 7.6 IC50 ChEMBL;BindingDB