Molecule Details
InChIKeyFQVCSBNTPQDQSS-UHFFFAOYSA-N
Compound NameN-[3-(4-hydroxycyclohexyl)oxynaphthalen-2-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
Canonical SMILESO=C(Nc1cc2ccccc2cc1OC1CCC(O)CC1)c1cnn2cccnc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.4
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9NWZ3 IRAK4 Homo sapiens Human PF07714 6.9 IC50 ChEMBL;BindingDB
P43405 SYK Homo sapiens Human PF07714 PF00017 6.2 IC50 ChEMBL;BindingDB
P51617 IRAK1 Homo sapiens Human PF00531 PF00069 6.1 IC50 ChEMBL;BindingDB