Molecule Details
InChIKeyFPVFNTHWCRWGPI-UHFFFAOYSA-N
Compound Name6-[(4-Cyano-phenyl)-thiazol-5-yl-methoxymethyl]-1-methyl-2-oxo-5-(4-trifluoromethoxy-phenyl)-1,2-dihydro-pyridine-3-carbonitrile
Canonical SMILESCn1c(COC(c2ccc(C#N)cc2)c2cncs2)c(-c2ccc(OC(F)(F)F)cc2)cc(C#N)c1=O
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL8.0
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 8.0 pIC50 TTD_MultiTarget
P49356 FNTB Homo sapiens Human PF00432 8.0 IC50 ChEMBL