Molecule Details
InChIKeyFPUIOUHUIOAZBC-CVEARBPZSA-N
Compound Name2-[(3R)-3-[[(2S)-2-benzyl-3-sulfanylpropanoyl]amino]-4-oxo-2,3-dihydro-1,5-benzothiazepin-5-yl]acetic acid
Canonical SMILESO=C(O)CN1C(=O)[C@@H](NC(=O)[C@@H](CS)Cc2ccccc2)CSc2ccccc21
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL8.38
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P08473 MME Homo sapiens Human PF01431 PF05649 9.0 IC50 ChEMBL;BindingDB
P12821 ACE Homo sapiens Human PF01401 7.8 IC50 ChEMBL;BindingDB