Molecule Details
InChIKeyFORMHTPKYXAYSB-SPHURBIESA-N
Compound Name(2S,4S)-N-[(1S)-2-(benzylamino)-2-oxo-1-propan-2-ylsulfanylethyl]-4-hydroxy-4-[(13S)-18-[methyl(methylsulfonyl)amino]-2,15-dioxo-4-phenyl-11-oxa-3,14-diazatricyclo[14.3.1.15,9]henicosa-1(19),5,7,9(21),16(20),17-hexaen-13-yl]-2-propan-2-ylbutanamide
Canonical SMILESCC(C)S[C@H](NC(=O)[C@@H](C[C@H](O)[C@@H]1COCc2cccc(c2)C(c2ccccc2)NC(=O)c2cc(cc(N(C)S(C)(=O)=O)c2)C(=O)N1)C(C)C)C(=O)NCc1ccccc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.02
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P07339 CTSD Homo sapiens Human PF07966 PF00026 9.1 Ki ChEMBL;BindingDB
P00797 REN Homo sapiens Human PF07966 PF00026 8.3 Ki ChEMBL;BindingDB
P56817 BACE1 Homo sapiens Human PF00026 6.6 IC50 ChEMBL;BindingDB