Molecule Details
InChIKeyFOMUZVDWSAHVBW-UHFFFAOYSA-N
Compound Name4-(3,4-Difluoro-phenyl)-3-{3-[4-(2-ethoxy-phenyl)-piperazin-1-yl]-propylcarbamoyl}-6-methyl-2-oxo-1,2,3,4-tetrahydro-pyrimidine-5-carboxylic acid methyl ester
Canonical SMILESCCOc1ccccc1N1CCN(CCCNC(=O)N2C(=O)NC(C)=C(C(=O)OC)C2c2ccc(F)c(F)c2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.64
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P35348 ADRA1A Homo sapiens Human PF00001 10.0 Ki ChEMBL;BindingDB
P35368 ADRA1B Homo sapiens Human PF00001 8.1 Ki ChEMBL;BindingDB
P25100 ADRA1D Homo sapiens Human PF00001 7.8 Ki ChEMBL;BindingDB