Molecule Details
InChIKeyFMZKGKLLLCYGJW-QWXGXRTQSA-N
Compound Name[(3R,4S)-6-(3-chloro-1H-indol-7-yl)-5,7-difluoro-2,2,4-trimethyl-3,4-dihydro-1H-quinolin-3-yl] N-benzylcarbamate
Canonical SMILESC[C@H]1c2c(cc(F)c(-c3cccc4c(Cl)c[nH]c34)c2F)NC(C)(C)[C@@H]1OC(=O)NCc1ccccc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.79
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P04150 NR3C1 Homo sapiens Human PF02155 PF00104 PF00105 7.4 IC50 ChEMBL;BindingDB
P06401 PGR Homo sapiens Human PF00104 PF02161 PF00105 6.8 Ki ChEMBL;BindingDB
P08235 NR3C2 Homo sapiens Human PF00104 PF00105 6.2 Ki ChEMBL;BindingDB