Molecule Details
InChIKeyFMQWOAKTQPLQBR-SANMLTNESA-N
Compound Name(5S)-5-(4-chlorophenyl)-N-[4-(4-fluorophenoxy)phenyl]-7,8-dihydro-5H-1,6-naphthyridine-6-carboxamide
Canonical SMILESO=C(Nc1ccc(Oc2ccc(F)cc2)cc1)N1CCc2ncccc2[C@@H]1c1ccc(Cl)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL6.51
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P22888 LHCGR Homo sapiens Human PF00001 PF13306 6.9 IC50 ChEMBL;BindingDB
P10632 CYP2C8 Homo sapiens Human PF00067 6.2 IC50 ChEMBL;BindingDB