Molecule Details
InChIKeyFMPNFDSPHNUFOS-HAHRSARXSA-N
Compound Name(3S,3aS,4R,4aS,8aS,9aR)-4-[(E)-2-[(2R,6S)-1,6-dimethylpiperidin-2-yl]ethenyl]-3-methyl-3a,4,4a,5,6,7,8,8a,9,9a-decahydro-3H-benzo[f][2]benzofuran-1-one
Canonical SMILESC[C@@H]1OC(=O)[C@@H]2C[C@@H]3CCCC[C@@H]3[C@@H](/C=C/[C@H]3CCC[C@H](C)N3C)[C@H]12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.72
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P08172 CHRM2 Homo sapiens Human PF00001 7.0 Ki ChEMBL;BindingDB
P08173 CHRM4 Homo sapiens Human PF00001 6.8 Ki ChEMBL;BindingDB
P11229 CHRM1 Homo sapiens Human PF00001 6.4 Ki ChEMBL;BindingDB