Molecule Details
InChIKeyFMMQGWSMYANLDD-VQHVLOKHSA-N
Compound Name3-methyl-5-(4-methyl-3-(3-((4-methylpiperazin-1-yl)methyl)styryl)-1H-indazol-5-yl)aniline
Canonical SMILESCc1cc(N)cc(-c2ccc3[nH]nc(/C=C/c4cccc(CN5CCN(C)CC5)c4)c3c2C)c1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.81
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q96GD4 AURKB Homo sapiens Human PF00069 7.5 IC50 ChEMBL;BindingDB
O14965 AURKA Homo sapiens Human PF00069 6.5 IC50 ChEMBL;BindingDB
O75716 STK16 Homo sapiens Human PF00069 6.5 pIC50 TTD_MultiTarget