Molecule Details
InChIKeyFMECAVUOMUCKKM-UHFFFAOYSA-N
Compound NameN-[3-[3-[[2-methyl-6-(3-morpholin-4-ylpropylamino)pyrimidin-4-yl]amino]-1H-pyrazol-5-yl]phenyl]benzenesulfonamide
Canonical SMILESCc1nc(NCCCN2CCOCC2)cc(Nc2cc(-c3cccc(NS(=O)(=O)c4ccccc4)c3)n[nH]2)n1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.78
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P36888 FLT3 Homo sapiens Human PF00047 PF07714 8.0 IC50 ChEMBL;BindingDB
O14965 AURKA Homo sapiens Human PF00069 6.2 IC50 ChEMBL;BindingDB
Q02161 RHD Homo sapiens Human PF00909 6.2 pIC50 TTD_MultiTarget