Molecule Details
InChIKeyFLYJDKQWLFTMBW-UHFFFAOYSA-N
Compound Name3-ethyl-1-(2-methoxyethyl)-5-methyl-6-[(2-oxo-1H-imidazol-3-yl)methyl]thieno[2,3-d]pyrimidine-2,4-dione
Canonical SMILESCCn1c(=O)c2c(C)c(Cn3cc[nH]c3=O)sc2n(CCOC)c1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.26
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P29275 ADORA2B Homo sapiens Human PF00001 8.6 Ki ChEMBL;BindingDB
P29274 ADORA2A Homo sapiens Human PF00001 7.0 Ki ChEMBL;BindingDB
P30542 ADORA1 Homo sapiens Human PF00001 6.2 Ki ChEMBL;BindingDB