Molecule Details
InChIKeyFLPMIYWQXAHVEM-UHFFFAOYSA-N
Compound Name6-[(3-Methoxy-5-trifluoromethylphenylamino)methyl]-2,4-diamino-5-methylpyrido[2,3-d]pyrimidine
Canonical SMILESCOc1cc(NCc2cnc3nc(N)nc(N)c3c2C)cc(C(F)(F)F)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.34
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00374 DHFR Homo sapiens Human PF00186 8.3 IC50 ChEMBL;BindingDB
O30463 folA Mycobacterium avium Pathogen PF00186 9.0 IC50 ChEMBL
Q07422 Toxoplasma gondii Pathogen PF00186 PF00303 7.7 IC50 ChEMBL;BindingDB