Molecule Details
InChIKeyFLGHEYRTVBXLCT-UHFFFAOYSA-N
Compound Name3-[4-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl]-5-phenyl-1,3,4-oxadiazol-2-one
Canonical SMILESCOc1cc2c(cc1OC)CN(CCCCn1nc(-c3ccccc3)oc1=O)CC2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.57
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q05586 GRIN1 Homo sapiens Human PF01094 PF00060 PF10613 7.6 Ki ChEMBL;BindingDB
Q13224 GRIN2B Homo sapiens Human PF01094 PF00060 PF10613 PF10565 7.6 Ki ChEMBL