Molecule Details
InChIKeyFKUAUADTVPZXDK-UHFFFAOYSA-N
Canonical SMILESCCn1c(N)nc2ccc(-c3cnc(OC)c(S(=O)(=O)Nc4ccc(F)cc4F)c3)cc2c1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.1
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P42356 PI4KA Homo sapiens Human PF00454 PF00613 PF19274 7.4 IC50 ChEMBL;BindingDB
P48736 PIK3CG Homo sapiens Human PF00454 PF00792 PF00794 PF00613 PF19710 6.8 IC50 ChEMBL;BindingDB