Molecule Details
InChIKeyFKCNXNPZSKIRIX-UHFFFAOYSA-N
Compound Name1-[3-(2-Ethoxyethoxy)-5,5,8,8-tetramethyl-6,7-dihydronaphthalen-2-yl]-2-(trifluoromethyl)benzimidazole-5-carboxylic acid
Canonical SMILESCCOCCOc1cc2c(cc1-n1c(C(F)(F)F)nc3cc(C(=O)O)ccc31)C(C)(C)CCC2(C)C
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.9
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P37231 PPARG Homo sapiens Human PF00104 PF12577 PF00105 7.2 Kd ChEMBL
Q13133 NR1H3 Homo sapiens Human PF00104 PF00105 6.8 Kd ChEMBL
P19793 RXRA Homo sapiens Human PF00104 PF11825 PF00105 6.8 Kd ChEMBL;BindingDB