Molecule Details
InChIKeyFKCNGHIFFXLRHA-JTQLQIEISA-N
Compound NameUS11066396, Example 105
Canonical SMILESCCc1nnc([C@@H]2CCC(=O)N2c2cc(F)c(-c3noc(C(F)(F)F)n3)cc2F)o1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.3
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9UBN7 HDAC6 Homo sapiens Human PF00850 PF02148 8.0 IC50 ChEMBL;BindingDB
Q9UQL6 HDAC5 Homo sapiens Human PF12203 PF00850 7.7 IC50 ChEMBL;BindingDB
Q13547 HDAC1 Homo sapiens Human PF00850 6.2 IC50 ChEMBL;BindingDB