Molecule Details
InChIKeyFKCMDMVCVNAORO-UHFFFAOYSA-N
Canonical SMILESCCCc1nc(CC)c(C(=O)OCc2ccc(C(=O)N(c3ccccc3)c3ccccc3)cc2)n1Cc1ccc(-c2ccccc2-c2nn[nH]n2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.2
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P30556 AGTR1 Homo sapiens Human PF00001 7.7 IC50 ChEMBL;BindingDB
P50052 AGTR2 Homo sapiens Human PF00001 6.7 IC50 ChEMBL;BindingDB