Molecule Details
InChIKeyFKBQPAXZYUEULP-UHFFFAOYSA-N
Compound NameN-(2-(1H-1,2,4-triazol-3-yl)thiophen-3-yl)-2-(naphthalen-1-yl)acetamide
Canonical SMILESO=C(Cc1cccc2ccccc12)Nc1ccsc1-c1nc[nH]n1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.16
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P45983 MAPK8 Homo sapiens Human PF00069 6.3 IC50 ChEMBL;BindingDB
P53779 MAPK10 Homo sapiens Human PF00069 6.0 IC50 ChEMBL;BindingDB