Molecule Details
InChIKeyFJSKRKLUQFIKJP-HWFRFQLBSA-N
Compound Name(S)-2-[(S)-4-{(R)-2-[(S)-2-acetylamino-3-(3H-imidazol-4-yl)-propionylamino]-3-phenyl-propionyl}-3-(3-guanidino-propyl)-2-oxo-piperazin-1-yl]-N-methyl-3-naphthalen-2-yl-propionamide
Canonical SMILESCNC(=O)[C@H](Cc1ccc2ccccc2c1)N1CCN(C(=O)[C@@H](Cc2ccccc2)NC(=O)[C@H](Cc2c[nH]cn2)NC(C)=O)[C@@H](CCCN=C(N)N)C1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.17
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q01726 MC1R Homo sapiens Human PF00001 9.4 Ki ChEMBL;BindingDB
P32245 MC4R Homo sapiens Human PF00001 9.1 Ki ChEMBL;BindingDB
P41968 MC3R Homo sapiens Human PF00001 9.0 Ki ChEMBL;BindingDB