Molecule Details
InChIKeyFIUCLBJMUGCQTF-LLVKDONJSA-N
Compound Name6-[[(1R)-1-(4-chlorophenyl)ethyl]amino]-1-cyclopentyl-5H-pyrazolo[5,4-d]pyrimidin-4-one
Canonical SMILESC[C@@H](Nc1nc2c(cnn2C2CCCC2)c(=O)[nH]1)c1ccc(Cl)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.81
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O76083 PDE9A Homo sapiens Human PF00233 7.2 IC50 ChEMBL
Q01064 PDE1B Homo sapiens Human PF00233 PF08499 7.1 IC50 ChEMBL
O76074 PDE5A Homo sapiens Human PF01590 PF00233 6.1 IC50 ChEMBL