Molecule Details
InChIKeyFIRZNFNHYVXQPP-IBGZPJMESA-N
Compound Name2-(2-chloro-N-[6-[4-[(2S)-3-(dimethylamino)-2-hydroxypropoxy]anilino]pyrimidin-4-yl]-5-methylanilino)acetonitrile
Canonical SMILESCc1ccc(Cl)c(N(CC#N)c2cc(Nc3ccc(OC[C@@H](O)CN(C)C)cc3)ncn2)c1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.09
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P11802 CDK4 Homo sapiens Human PF00069 7.3 IC50 ChEMBL
P24941 CDK2 Homo sapiens Human PF00069 6.8 pIC50 TTD_MultiTarget