Molecule Details
InChIKeyFHVZRKFXAWGVLU-UHFFFAOYSA-N
Compound Name(+/-)-4-Benzo[b]thiophen-5-yl-2-methyl-7-pyridazin-3-yl-1,2,3,4-tetrahydroisoquinoline
Canonical SMILESCN1Cc2cc(-c3cccnn3)ccc2C(c2ccc3sccc3c2)C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.53
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P23975 SLC6A2 Homo sapiens Human PF00209 8.8 Ki ChEMBL;BindingDB
P31645 SLC6A4 Homo sapiens Human PF03491 PF00209 8.7 Ki ChEMBL;BindingDB
Q01959 SLC6A3 Homo sapiens Human PF00209 8.1 Ki ChEMBL;BindingDB