Molecule Details
InChIKeyFHTSRDNJZWDVBC-UHFFFAOYSA-N
Compound Name6-Ethyl-5-[3-(2-methoxy-5-phenylphenyl)but-1-ynyl]pyrimidine-2,4-diamine
Canonical SMILESCCc1nc(N)nc(N)c1C#CC(C)c1cc(-c2ccccc2)ccc1OC
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.25
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00374 DHFR Homo sapiens Human PF00186 7.0 IC50 ChEMBL;BindingDB
J7IFZ2 Streptococcus pyogenes Pathogen PF00186 7.6 IC50 ChEMBL;BindingDB
P0A017 folA Staphylococcus aureus Pathogen PF00186 7.2 IC50 ChEMBL;BindingDB