Molecule Details
InChIKeyFHSKCOBLBQSSQE-CMDGGOBGSA-N
Compound Name5-(pyridin-4-yl)-6-(pyrrolidin-1-yl)-3-styryl-1H-indazole
Canonical SMILESC(=C/c1n[nH]c2cc(N3CCCC3)c(-c3ccncc3)cc12)\c1ccccc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.98
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q96GD4 AURKB Homo sapiens Human PF00069 7.3 IC50 ChEMBL;BindingDB
O14965 AURKA Homo sapiens Human PF00069 6.8 IC50 ChEMBL;BindingDB
O75716 STK16 Homo sapiens Human PF00069 6.8 pIC50 TTD_MultiTarget