Molecule Details
InChIKeyFHILGPQALCJBPN-UHFFFAOYSA-N
Compound Name5-(12-Methoxy-5,7-dimethyl-2,4,8,13-tetrazatricyclo[7.4.0.02,6]trideca-1(9),3,5,7,10,12-hexaen-3-yl)-2,4-dimethyl-1,3-thiazole
Canonical SMILESCOc1ccc2nc(C)c3c(C)nc(-c4sc(C)nc4C)n3c2n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.34
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9Y233 PDE10A Homo sapiens Human PF01590 PF00233 8.4 IC50 ChEMBL;BindingDB
O00408 PDE2A Homo sapiens Human PF01590 PF00233 7.5 IC50 ChEMBL;BindingDB
Q13946 PDE7A Homo sapiens Human PF00233 6.1 IC50 ChEMBL;BindingDB