Molecule Details
InChIKeyFHESSCZVRQCSRX-KSSFIOAISA-N
Compound Nametrans-(1S,2S)-2-[6-(1-pyridin-2-ylpyrazolo[4,3-c]pyridin-6-yl)pyrazin-2-yl]oxycyclopentan-1-amine
Canonical SMILESN[C@H]1CCC[C@@H]1Oc1cncc(-c2cc3c(cn2)cnn3-c2ccccn2)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.77
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q86V86 PIM3 Homo sapiens Human PF00069 10.2 Ki ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 10.0 Ki ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 9.1 Ki ChEMBL;BindingDB