Molecule Details
InChIKeyFGLVLXDXUNBIQC-PFYATKOYSA-N
Compound Name(2Z,5R)-2-[(1-benzylindol-3-yl)methylidene]-3-oxo-N,5-diphenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
Canonical SMILESO=C(Nc1ccccc1)C1=CN=c2s/c(=C\c3cn(Cc4ccccc4)c4ccccc34)c(=O)n2[C@@H]1c1ccccc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)4
Pfam Stratification Cross-Family
Avg pChEMBL6.26
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (4)
Target Gene Organism Category Pfam pChEMBL Type Source
P55957 BID Homo sapiens Human PF06393 6.4 Ki ChEMBL
Q07820 MCL1 Homo sapiens Human PF00452 6.4 Ki ChEMBL
O43521 BCL2L11 Homo sapiens Human PF08945 PF06773 6.1 Ki ChEMBL
Q07817 BCL2L1 Homo sapiens Human PF00452 PF02180 6.1 Ki ChEMBL