Molecule Details
InChIKeyFGLLFRICMCXRAJ-HBBKIPDOSA-N
Compound Name(3R,5S)-1-[dideuterio(phenyl)methyl]-3,5-dimethyl-N-pyridin-3-yl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Canonical SMILES[2H]C([2H])(c1ccccc1)N1C[C@@H](C)N(C(=O)Nc2cccnc2)[C@@H](C)c2ccccc21
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.86
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9P0X4 CACNA1I Homo sapiens Human PF00520 8.4 IC50 ChEMBL;BindingDB
O95180 CACNA1H Homo sapiens Human PF00520 7.6 IC50 ChEMBL;BindingDB
O43497 CACNA1G Homo sapiens Human PF00520 7.6 IC50 ChEMBL;BindingDB