Molecule Details
InChIKeyFGDXJSBOTIKISM-RUZDIDTESA-N
Compound Name1-(3H-Imidazol-4-ylmethyl)-4-methanesulfonyl-7-phenyl-3-pyridin-3-ylmethyl-2,3,4,5-tetrahydro-1H-benzo[e][1,4]diazepine
Canonical SMILESCS(=O)(=O)N1Cc2cc(-c3ccccc3)ccc2N(Cc2c[nH]cn2)C[C@H]1Cc1cccnc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL8.23
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 8.2 pIC50 TTD_MultiTarget
P49356 FNTB Homo sapiens Human PF00432 8.2 IC50 ChEMBL;BindingDB