Molecule Details
InChIKeyFGBDLJIVZVBTAG-UHFFFAOYSA-N
Compound Name5-{2-[4-(3H-Benzimidazol-4-ylmethyl)piperazin-1-yl]ethoxy}-2-methylquinoline
Canonical SMILESCc1ccc2c(OCCN3CCN(Cc4cccc5[nH]cnc45)CC3)cccc2n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.87
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28221 HTR1D Homo sapiens Human PF00001 9.6 Ki ChEMBL;BindingDB
P28222 HTR1B Homo sapiens Human PF00001 7.2 Ki ChEMBL;BindingDB
P08908 HTR1A Homo sapiens Human PF00001 6.8 Ki ChEMBL;BindingDB