Molecule Details
InChIKeyFFBYNQCXDQNNQT-GKQHHHCTSA-N
Canonical SMILESCc1c(NC[C@H]2CCC[C@@H](c3ccc(C(F)(F)F)cc3)O2)nc(C2CCOCC2)nc1C(=O)N1CCC(N[C@H]2CCOC[C@H]2F)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.84
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P41597 CCR2 Homo sapiens Human PF00001 9.0 Ki ChEMBL;BindingDB
P51681 CCR5 Homo sapiens Human PF00001 6.7 Ki ChEMBL;BindingDB