Molecule Details
InChIKeyFEWLFECITKFLDY-QUCCMNQESA-N
Compound Namecis-(1S,2R)-2-[[[7-(benzylamino)-3-propan-2-ylpyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]cyclohexan-1-ol
Canonical SMILESCC(C)c1cnn2c(NCc3ccccc3)cc(NC[C@H]3CCCC[C@@H]3O)nc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.16
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P50613 CDK7 Homo sapiens Human PF00069 6.2 IC50 ChEMBL;BindingDB
P51946 CCNH Homo sapiens Human PF16899 PF00134 6.2 IC50 ChEMBL;BindingDB
P51948 MNAT1 Homo sapiens Human PF25811 PF06391 PF17121 6.2 IC50 ChEMBL