Molecule Details
InChIKeyFEFCYILNMDAYPD-FQEVSTJZSA-N
Compound NameN-[2-[[2-[(2S)-2-cyanopyrrolidin-1-yl]-2-oxoethyl]amino]-2-methylpropyl]-5,7-dimethyl-2-phenylpyrazolo[1,5-a]pyrimidine-6-carboxamide
Canonical SMILESCc1nc2cc(-c3ccccc3)nn2c(C)c1C(=O)NCC(C)(C)NCC(=O)N1CCC[C@H]1C#N
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.72
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q6V1X1 DPP8 Homo sapiens Human PF19520 PF00930 PF00326 7.9 IC50 ChEMBL;BindingDB
Q86TI2 DPP9 Homo sapiens Human PF19520 PF00930 PF00326 7.7 IC50 ChEMBL;BindingDB
P27487 DPP4 Homo sapiens Human PF00930 PF00326 7.5 IC50 ChEMBL;BindingDB