Molecule Details
InChIKeyFECGNZAYTJHJIY-UHFFFAOYSA-N
Compound Name4-methyl-N-[4-[(1-methylpiperidin-4-yl)methoxy]-3-(trifluoromethyl)phenyl]-3-[[1-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)cyclopropanecarbonyl]amino]benzamide
Canonical SMILESCc1ccc(C(=O)Nc2ccc(OCC3CCN(C)CC3)c(C(F)(F)F)c2)cc1NC(=O)C1(c2ncnc3[nH]ccc23)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.21
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P15056 BRAF Homo sapiens Human PF00130 PF07714 PF02196 7.4 IC50 ChEMBL;BindingDB
P04049 RAF1 Homo sapiens Human PF00130 PF07714 PF02196 7.2 IC50 ChEMBL;BindingDB
P10398 ARAF Homo sapiens Human PF00130 PF07714 PF02196 7.0 IC50 ChEMBL;BindingDB