Molecule Details
InChIKeyFDWJEDYUZLTROC-UHFFFAOYSA-N
Compound Name3-[2-(2-aminopyrimidin-5-yl)ethynyl]-N-[3-(trifluoromethyl)phenyl]benzamide
Canonical SMILESNc1ncc(C#Cc2cccc(C(=O)Nc3cccc(C(F)(F)F)c3)c2)cn1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.36
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q02763 TEK Homo sapiens Human PF00041 PF10430 PF07714 9.0 pIC50 TTD_MultiTarget
P06239 LCK Homo sapiens Human PF07714 PF00017 PF00018 7.7 IC50 ChEMBL;BindingDB