Molecule Details
InChIKeyFCAIKTYDWLTVQR-UHFFFAOYSA-N
Compound Name7-Bromo-3-(3-chloro-benzyl)-1-(3H-imidazol-4-ylmethyl)-4-methanesulfonyl-2,3,4,5-tetrahydro-1H-benzo[e][1,4]diazepine
Canonical SMILESCS(=O)(=O)N1Cc2cc(Br)ccc2N(Cc2c[nH]cn2)CC1Cc1cccc(Cl)c1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.62
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 7.6 pIC50 TTD_MultiTarget
P49356 FNTB Homo sapiens Human PF00432 7.6 IC50 ChEMBL;BindingDB