Molecule Details
InChIKeyFBBVGKUOXFKGAI-GUIRCDHDSA-N
Compound Name4-sulfamoyl-N-({1-[(2R,3S,4R,5R)-3,4,5-trihydroxyoxan-2-yl]-1H-1,2,3-triazol-4-yl}methyl)benzamide
Canonical SMILESNS(=O)(=O)c1ccc(C(=O)NCc2cn([C@@H]3OC[C@@H](O)[C@@H](O)[C@@H]3O)nn2)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.72
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00918 CA2 Homo sapiens Human PF00194 6.9 Ki ChEMBL;BindingDB
P18505 GABRB1 Homo sapiens Human PF02931 PF02932 6.9 pIC50 TTD_MultiTarget
Q16790 CA9 Homo sapiens Human PF00194 6.4 Ki ChEMBL;BindingDB